Naphthyridine containing antibacterial agent
Witryna2 cze 2010 · A large number of 1,8-naphthyridine derivatives are reported to exhibit antibacterial, antimalarial 9 and anticancer 10 activities. Our earlier studies also have … WitrynaA series of 7,8-disubstituted 1-cyclopropyl-6-fluoroquinoline-3-carboxylic acids, 7-substituted 1-cyclopropyl-6-fluoro-1,8-naphthyridine-3-carboxylic acids, and 10-substituted 9-fluoropyridobenzoxazine-6-carboxylic acids has been prepared and evaluated for antibacterial activity. The side chains exa …
Naphthyridine containing antibacterial agent
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Witryna15 lip 2012 · 7.15.12 Important Compounds and Applications. Medicinally important naphthyridine derivatives such as analogues of the antibacterial agent naladixic … Witryna1 lut 2024 · The silver(I) complexes with 1,5-naphthyridine (1,5-naph), Ag1–3, were prepared in a good yield (~70%) by reacting 1,5-naph with an equimolar amount of …
Witryna20 gru 2024 · Nalidixic acid is the first 4‐quinolone antibacterial agent with α, β unsaturated carboxylic acid at the 2, 3 positions of the 1,8 naphthyridine nucleus (Assaleh, Chandu, Peraman, & Katakam, 2013; Nicolle, 2005). Following oral administration, nalidixic acid failed to achieve optimum plasma or tissue … WitrynaThere are disclosed new naphthyridine- and quinoline-carboxylic acids having a 1-tertiary-alkyl substituent, compositions containing them, and their use in treating bacterial infections in warm-blooded animals. Also disclosed are novel amines and intermediates used in the preparation of the naphthyridine- and quinoline-carboxylic …
Witryna6 gru 2024 · Nitrogen-containing heterocycles such as 1,8-naphthyridine derivatives have been shown to have excellent antimicrobial properties. Therefore, the purpose … Witryna1 lut 1990 · New quinolone antibacterial agents. Synthesis and biological activity of 7-(3,3- or 3,4-disubstituted-1-pyrrolidinyl)quinoline-3-carboxylic acids. Susan E. Hagen, …
WitrynaThe article was published on 1989-07-25. It has received 25 citation(s) till now. The article focuses on the topic(s): Substituent & Side chain.
WitrynaThe search for new antibacterial agents has become urgent due to the exponential growth of bacterial resistance to antibiotics. Nitrogen-containing heterocycles such as 1,8-naphthyridine derivatives have been shown to have excellent antimicrobial properties. Therefore, the purpose of this study was to evaluate the antibacterial and … pembroke ga city hallWitrynaM. Y. Saleh et al. / Synthesis of Some Novel 1,8-Naphthyridine Chalcones activities and used as analgesics, antiviral, anti-inflammatory agent, antibacterial and anti-tuberculosis agent [10-12]. As well as its proposal as a drug against the emerging corona virus, by studying a theory using the Docking program [13]. mechatronics mcmasterWitrynaThere are disclosed new naphthyridine-and quinoline-carboxylic acids having a 1-tertiary-alkyl substituent, compositions containing them, and their use in treating bacterial infections in warm-blooded animals. Also disclosed are novel amines and intermediates used in the preparation of the naphthyridine-and quinoline-carboxylic … mechatronics model uf25gca12 bthWitryna1, 8- Naphthyridine nucleus belongs to significant nitrogen-containing heterocyclic compounds which has garnered the interest of researchers due to its versatile … pembroke flag football leagueWitrynaantibacterial agent Prior art date 1987-08-21 Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis … mechatronics md1238x24bWitrynaantibacterial agent naphthyridine derivatives naphthyridine Prior art date 1992-07-15 Application number SK46-95A Other languages English (en) Slovak (sk) Inventor ... C07D471/02 — Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, ... mechatronics melchett roadWitryna24 paź 1997 · New pyrrolidine derivatives, which bear an alkyloxime substituent in the 4-position and an aminomethyl substituent in the 3-position of the pyrrolidine ring, have been synthesized and coupled with various quinolinecarboxylic acids to produce a series of new fluoroquinolone antibacterials. These fluoroquinolones were found to possess … mechatronics md1238h12b